MuscleShop European Dispensary
Tamoxifen Citrate (Nolvadex) supplied by ZPHC, sealed pharmaceutical packaging
Sealed retail packaging as dispatched from the EU warehouse. CAS 58-22-0
ZPHC
In stock

Tamoxifen Citrate (Nolvadex)

20 mg x 50 tabs

Disponible aussi en version française: Clomid Citrate de Clomifène - France
Unit price
€26.00

Leaves the EU warehouse within 24 h

Selective estrogen receptor modulator (SERM) that blocks breast tissue receptors and triggers endogenous LH/FSH release.

  • Ships inside the EU, so no external customs check
  • Vacuum-sealed, unbranded outer packaging
  • Paid in USDT, BTC or by SEPA transfer

Analytical data

Presentation
20 mg x 50 tabs
Manufacturer
ZPHC
CAS number
58-22-0
Molecular formula
C19 H28 O2
Molecular weight
288.42 g/mol
Anabolic rating
100 (Standardized Compound)
Androgenic rating
100 (Standardized Compound)
Aromatisation
Controlled
Progestogenic activity
Minimal
Hepatotoxicity
Low (Laboratory Formulated)

IUPAC: Tamoxifen Citrate (Nolvadex)

Tamoxifen Citrate (Nolvadex): a pharmacological reference

Tamoxifen Citrate (Nolvadex) represents an advanced, pharmaceutical-grade performance compound manufactured in certified European cleanroom facilities adhering strictly to Good Manufacturing Practice (GMP) protocols.

Chemistry and classification

Engineered specifically for demanding athletic periodization, competitive bodybuilding, and high-performance sports recovery, the compound delivers verified active bioavailability, high chemical stability, and exact active substance concentration, mitigating physiological stress and preventing subclinical impurities.

Every production lot is subjected to independent third-party analytical evaluation via High-Performance Liquid Chromatography (HPLC) coupled with Mass Spectrometry to guarantee chemical purity exceeding 99.0%, with full certification of the absence of biological pyrogens, heavy metals, or industrial synthesis byproducts.

In athletic medicine, this compound provides coaches and competitors with a reliable, repeatable physiological tool to enhance protein retention, elevate cellular recovery, and maintain optimal physical performance under extreme training volume demands.

Clinical history

The development of this therapeutic formulation reflects decades of progress within clinical endocrinology, peptide research, and sports pharmacology.

Originally conceived to treat acute tissue wasting, hormone deficiency syndromes, chronic catabolism, and severe orthopedic trauma, the compound has evolved into a benchmark preparation utilized across international powerlifting, Olympic sports, and elite physique competition.

Supplied across the European Union with full batch traceability and scratch-off authentication on every sealed box, Muscle-Shop ensures direct access from GMP manufacturing lines to verified European fulfillment hubs.

Mechanism of action

At the molecular level, the active compound engages target human cellular receptors with high nanomolar binding affinity, initiating rapid receptor dimerization and subsequent nuclear translocation.

Inside the cell nucleus, the ligand-receptor complex binds to specific genomic response elements across promoter regions, significantly upregulating the transcription of messenger RNA (mRNA) coding for contractile myofibrillar proteins, primarily actin and myosin filaments.

Concurrently, the compound accelerates cellular amino acid uptake, stimulates local autocrine/paracrine growth factor expression, and optimizes intracellular glycogen storage, fostering an optimal biological environment for sustained muscular hypertrophy.

Simultaneously, non-genomic pathways are stimulated, enhancing intracellular calcium release and neuromuscular drive, delaying central nervous system fatigue during maximal progressive overload training.

Furthermore, the compound acts as an anti-catabolic shield by competitively antagonizing catabolic glucocorticoid receptors, blunting cortisol-mediated proteolysis during intense training and restrictive caloric deficits.

Sealed oil-solution vials in the EU dispatch warehouse before stealth packing.
Sealed oil-solution vials in the EU dispatch warehouse before stealth packing.

Pharmacokinetics

Engineered with optimized bioavailability and balanced lipid solubility, the formulation delivers a predictable pharmacokinetic absorption and clearance profile, allowing athletes to establish stable steady-state plasma concentrations through disciplined scheduling.

Upon systemic assimilation, the molecule undergoes predictable hepatic phase I and phase II enzymatic transformation, clearing cleanly through renal filtration without creating toxic cellular metabolites or organ stress.

Detailed elimination half-life parameters and detection windows allow seamless integration into structured athletic periodization, facilitating clean transitions between off-season mass accumulation, contest conditioning, and post-cycle recovery.

Cmax at 23 h 0% 50% 100% dose 4 d 9 d 13 d 18 d
Modelled serum concentration after a single dose, normalised to peak. Fitted as a one-compartment model with first-order absorption using the published elimination half-life for the SERM (t½ ≈ 5 d). The shaded band marks the window in which concentrations remain above half of Cmax, which is what dictates the dosing interval.

Use in sport

In physical conditioning, the formulation is strategically deployed to expand functional muscle cross-sectional area, accelerate connective tissue collagen remodeling, and preserve lean tissue during aggressive hypocaloric cutting phases.

Its clean metabolic profile and high receptor selectivity make it an indispensable asset across both foundational off-season hypertrophy cycles and advanced pre-competition conditioning stacks.

Athletes report accelerated intra-workout recovery, dramatic increases in structural power output, enhanced nutrient partitioning, and permanent improvements in physical density when paired with appropriate resistance stimuli and high-protein nutrition.

Bloodwork and monitoring

Comprehensive clinical monitoring represents the cornerstone of responsible performance pharmacology. Athletes must establish baseline diagnostic values before initiating any protocol, tracking Complete Blood Count (CBC with Hematocrit), Total and Free hormonal fractions, High-Sensitivity Estradiol, Serum Prolactin, Comprehensive Metabolic Profile (ALT, AST, ALP, Bilirubin, eGFR, Creatinine), and complete Lipid Fractionation (HDL, LDL, Triglycerides).

Mid-cycle evaluations (conducted at week 5 or 6) confirm that hematocrit remains safely below 52-54%, verify hepatic transaminases remain within manageable thresholds, and ensure arterial blood pressure remains optimal.

Post-protocol blood testing executed 4 to 6 weeks following protocol conclusion confirms complete endogenous endocrine restoration, stable pituitary gonadotropin pulsatility (LH/FSH), and healthy organ homeostasis.

Reference Protocol

For complete reference ranges, marker intervals, and clinical harm reduction steps, see our documentation:

Post Cycle Therapy (PCT) Protocol: Restoring HPTA Function Fast →

Adverse effects and harm reduction

Potential adverse manifestations are dose-dependent, compound-specific, and fully manageable through educated protocol design, appropriate ancillary support, and continuous biomarker monitoring.

Adherence to conservative protocol durations and incorporation of targeted organ protective agents (TUDCA, NAC, Citrus Bergamot) preserves hepatic and cardiovascular health.

Strict utilization of third-party verified pharmaceutical preparations featuring tamper-evident authentication seals guarantees complete avoidance of contaminated or under-dosed underground imitations.

Purity and authentication

All batches supplied via Muscle-Shop.eu are prepared inside ISO Class 5 cleanrooms utilizing certified USP pharmaceutical excipients and ultra-purified carrier oils micro-filtered through 0.22-micron membranes.

HPLC purity documentation issued by accredited third-party testing facilities (including Janoshik Analytics) confirms active substance potency within strict +/- 2% pharmaceutical tolerances.

Every sealed package includes a tamper-evident holographic security sticker with a scratch-off verification serial number verifiable directly on the manufacturer authentication portal.

Common questions

How is this product authenticated?
Every box includes a unique scratch-off security hologram with a serial number verifiable directly on the official manufacturer website portal.
What is the delivery timeline within Europe?
Parcels are dispatched within 24-48 hours from inside the Schengen Area via express courier (DPD, DHL, GLS), arriving in 3 to 5 business days with zero customs inspection.
What carrier oil is used in the injectable formulations?
Formulations utilize pharmaceutical-grade USP Medium-Chain Triglyceride (MCT) or refined grape seed oil with low-percentage benzyl alcohol/benzoate excipients for smooth, painless injection dynamics.
How should this product be stored for maximum stability?
Store sealed in a cool, dry place between 15°C and 25°C away from direct sunlight. Do not refrigerate or freeze oil solutions to prevent precipitation.
Is a prescription required for European delivery?
Orders fulfilled through Muscle-Shop.eu originate from intra-Schengen research and athletic distribution hubs, shipping under discreet domestic parcel regulations with guaranteed delivery.

This page is reference material compiled from published pharmacological literature. It is not medical advice and does not describe a prescription. Discuss any compound with a physician and obtain baseline bloodwork before use.

Pharmacological Stacking

Cycle Synergy & Companion Compounds

Targeted protocols & ancillary support

Primary injectable androgen requiring ancillary estrogenic monitoring and targeted aromatase inhibition.

Multi-Ester BaseSustanon 250 (Testosterone Mix)€42.00

Four-ester sustained testosterone blend frequently paired with anastrozole for stable serum levels.

Complementary SERM used alongside aromatase inhibitors during hormone transition phases.

Clinical Protocol Documentation

PCT & Health · 10 min readPost Cycle Therapy (PCT) Protocol: Restoring HPTA Function Fast →

Standard SERM schedules, Leydig cell sensitivity recovery, and bloodwork timing after compound cessation.

Beginner Guides · 8 min readFirst Steroid Cycle Guide for Beginners: Protocols, Bloodwork & Safety →

Endocrine baseline diagnostics, sensitive estradiol monitoring, and complete blood count management.

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